YM 254890 Size:2mg solid 5 h and oral bioavailability

Name: YM 254890 Size:2mg solid 5 h and oral bioavailability
Brand: pretereo.com
SKU: 38078312790
Price: 1079.92 USD
Availability: InStock
Rating: 4.4689000000000005 (10 reviews)

SKU: 38078312790

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Description

5 h and oral bioavailability of 100%

In xenograft models

esomeprazole

44)45)54-35(30)55-64(4

YM 254890 Size:2mg solid 5 h and oral bioavailabilityG protein inhibitor. Potently inhibits Gq 11 heterotrimeric G protein signaling. Inhibits ATP UTP induced Ca2+ increase in HCAE cells expressing P2Y2 receptor (IC50 = 50 nM); carbachol induced production of IP1 in CHO cells expressing M1 receptor (IC50 = 95 nM); and ADP induced Ca2+ increase in platelets, in vitro (IC50 = 2 M). Also inhibits Gs induced cAMP elevation and G protein coupled MAPK ERK signaling. Product information CAS Number: 568580 02 9

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